The drug 'Anaprilin': indications for use

The drug "Anaprilin" refers to the group of synthetic adrenoblockers used for the therapy of cardiac dysfunction, as well as under increased pressure.

The drug "Anaprilin": indications for use and pharmacological action

The work of the drug is to block the adrenoreceptors. Due to the effect of the drug, the oxygen demand of the myocardium, cardiac output, contractile work of the cardiac muscle decreases. With the help of medication, blood pressure decreases, peripheral resistance of blood vessels increases.

According to reviews and medical observations, the drug has an antiarrhythmic effect, raises the tone of the bronchi, increases uterine contractions, reduces the birth and post-operative bleeding.

The drug is quickly absorbed and removed from the human body. Half-life occurs after 4 hours, with prolonged admission - after 12 hours. The bulk of the drug goes through the kidneys as metabolites, and only one percent of the drug is excreted unchanged.

The drug "Anaprilin": indications for use and form of release

The drug is produced in the form of tablets and in ampoules. In the first case, the medicine is released at 1 and 4 milligrams in packs of 10, 50 and 100 units. The injection solution goes on sale at 0.25% (in 1 milliliter) and 0.1% (in 1 and 5 ml).

The drug is prescribed for the treatment of angina, heart rhythm disorders associated with rheumatoid lesions (sinus and paroxysmal tachycardia, arrhythmia, extrasystole, ciliary tachyarrhythmia). The medicine is used for hypertension, thyrotoxicosis, pheochromocytoma, ischemic heart disease.

The drug Anaprilin: how to take

The necessary dose for treatment is prescribed by the doctor. Usually in the form of a solution for injection, the drug is administered three to four times a day for 10 mg per quarter of an hour before meals. If the proper effect does not occur, these doses are gradually increased to 20 ... 40 mg.

For arrhythmia therapy, a 10-30 mg dose is indicated according to the above scheme. With angina in the first three days, 20 mg of the drug are taken four times, 40 mg for the next three days. On the fourth day 20 mg are prescribed, and from the seventh day the medicine is given four times 40 mg each.

Intramuscularly, a 1% solution of the drug is prescribed with open-angle glaucoma to reduce intraocular pressure. Intravenous use is carried out for violations of the heart rate and for the suppression of angina attacks.

Strict medical indications do not exclude the administration of the drug to children. In such cases, the medicine is given at the rate of a quarter to half a milligram per kilogram of the child's weight.

The drug Anaprilin: indications for use and side effects

During treatment, such negative manifestations as nausea, vomiting, diarrhea, deterioration of sleep, general weakness and dizziness are possible. Side effects also include hypotension, bradycardia; Itching can occur, symptoms of insufficient blood circulation, with long-term use impotence occurs. Side effects also occur with individual intolerance of the drug.

The drug Anaprilin: indications for use and contraindications

Doctors forbid taking medicine during an exacerbation of myocardial infarction, with bronchial asthma, diabetes, when peripheral arterial blood flow disturbances occur. The drug is contraindicated for such abnormalities as spastic colitis, sinus bradycardia, hay fever, complete and incomplete atrioventricular block, predisposition to bronchospasm. Only in extreme cases is prescribed the drug "Anaprilin" during pregnancy and during the feeding of the child.