HealthPreparations

"Relaxon" preparation: instructions for use, description, reviews, analogues

In what dose do they prescribe the drug Relaxon? Instructions for use of the medicament will be discussed below. Also you will learn about whether there are analogues for this medicine, how much it costs, in what cases it is not prescribed, etc.

Form, description, composition and packaging

The preparation "Relaxon" is produced in the form of round biconvex tablets of white color, covered with a film membrane. The active substance of this drug is zopiclone. Also in the composition of the medicament are the following auxiliary substances: methyloxypropylcellulose, microcrystalline cellulose, lactose, potato starch, colloidal silicon dioxide, talc, sodium carboxymethyl starch, povidone, macrogol, magnesium stearate and titanium dioxide.

In what kind of packaging are the tablets "Relaxon" sold? Instructions for use are enclosed in a pack of cardboard, where the contour cells with the drug are placed.

Pharmacodynamic characteristics

How does the drug "Relaxon" work? Instruction for use reports that this is a hypnotic, belonging to a group of cyclopirrolone. Structurally, it differs from barbiturates and hypnotic benzodiazepine series. This drug is a benzodiazepine receptor agonist. Interacting with them, it does not come into contact with peripheral receptors.

Properties of the preparation

What are the properties of the "Relaxon" medication? Experts say that this tool is able to have sedative, moderate anticonvulsant sleeping pills, muscle relaxant and tranquilizing effects. All of them are related to the action from the receptors of the macromolecular complex GABA.

After taking the pill, the inhibitory effect of GABA is increased, and the inter-neural transmission in the central nervous system is suppressed.

Sleeping "Relaxon" significantly shortens the time of falling asleep, reduces the number of awakenings at night and improves the quality of sleep. Also this drug prolongs the duration of sleep and almost does not cause such post-somnical effects as drowsiness and malaise in the morning.

Adapting to the action of the drug is absent. Therefore, it can be taken in a batch mode up to 17 weeks.

Pharmacokinetics of the drug

The drug "Relaxon", the price of which is indicated below, is quickly absorbed and is observed in the blood after 2 hours. The intake of food does not affect the absorption of the drug in any way. At 45%, it binds to blood proteins.

Even after several pills, the accumulation of their active substance, as well as metabolites, is not observed.

The half-life of zopiclone and the main metabolites is 7.5 and 4.5 hours, and the unchanged zopiclone is 5.5 hours. Approximately 80% of the drug is excreted together with urine, and 17-20% with feces.

In elderly people, the metabolism of the drug in the liver is somewhat reduced. At the same time, its half-life is extended to 7 hours. As for the accumulation of the active substance, then with repeated administration of tablets, it is not detected.

Indications for use

What to do with insomnia? Doctors recommend taking "Relaxon". This drug is designed to treat chronic, situational and transient insomnia in adults. Also it is actively used by those who have difficulty with falling asleep, early and night awakenings.

Contraindications for use

Tablets "Relaxon" is not recommended for taking in the following cases:

  • With increased sensitivity to the main substance of the drug;
  • With severe myasthenia gravis;
  • During pregnancy;
  • Sleep apnea ;
  • With respiratory failure;
  • With severe hepatic insufficiency;
  • Under the age of 18 years.

"Relaxon" preparation: instructions for use

Before taking a hypnotic, it is recommended to consult a doctor. Also it is necessary to study the enclosed instruction.

Tablets "Relaxon" (international name - "Zopiclone") are taken orally, shortly before the onset of sleep. Adults receive this medication at a dose of 7.5 mg. The maximum amount of sleeping pills is 15 mg.

The total duration of the use of tablets should not be more than one month. In each individual case, the duration of therapy is determined individually, depending on the patient's condition and the form of insomnia.

It is desirable to take the drug with transient insomnia about 3-5 days, and for a situational one - 2.5-3 weeks. The duration of the course therapy of chronic insomnia should be determined only by the doctor.

Elderly people with chronic pulmonary insufficiency, as well as with impaired liver function, are prescribed 3.75 mg of the drug. If necessary, this dosage can be increased to 7.5 mg.

The treatment of insomnia in patients with kidney failure also begin with ½ tablets, that is, with 3.75 mg.

Cases of overdose

Taking large doses of a hypnotic causes CNS depression of varying severity (from pronounced drowsiness to a coma).

The overdose therapy starts with a gastric lavage. Then the patient is assigned sorbents.

Symptomatic treatment and monitoring of vital body functions is also carried out. The drug "Flumazenil" is used as an antidote.

Side effects

What are the side effects of Relaxon? The responses of experienced specialists say that this medication can contribute to the development of the following phenomena:

  • Nausea, dryness and bitterness in the mouth;
  • Dizziness, headache, mild drowsiness in the morning;
  • Nightmares, aggressiveness, irritability, hallucinations, mood worsening and depressive state, as well as the development of amnesia (very rarely);
  • Itching, rash, anaphylactic reactions (extremely rare);
  • Increased transaminases of the liver and alkaline phosphatase.

It should also be noted that in rare cases, the drug causes the syndrome of "cancellation" and as a consequence, ricochet insomnia.

Drug Interactions

Now you know what to do with insomnia. Reception of the drug "Relaxon" should be extremely cautious, especially with the simultaneous use of other medications.

According to the attached instructions, the increase in the oppressive effect on the CNS of this drug occurs when combined with antidepressants, neuroleptics, anesthetics, tranquilizers, sedatives and hypnotics, as well as "Erythromycin", antiepileptic and antihistamines, narcotic analgesics.

It is highly not recommended to drink alcoholic drinks and alcohol-containing medicines at the same time as Relaxon. This is due to the fact that such a combination can enhance its sedative effect.

Taking a hypnotic drug significantly reduces the concentration of perforanal or trimipramine in the blood. This fact must be taken into account when they are simultaneously assigned.

Special recommendations for the taking of sleeping pills

What should I know before taking the drug Relaxon (analogues of this remedy are listed below)?

In people with night attacks of bronchial asthma in combination with medications of the methylxanthine series, the hypnotic reduces the number of attacks in the pre-hours, and also reduces their intensity and duration.

When appointing "Relaxon", one should not completely exclude the possibility of developing addiction. The risk of dependence on the drug occurs in the following cases:

  • If the duration of treatment and dosage is disturbed;
  • When drinking alcohol or other drugs;
  • When combined with alcohol or other psychotropic drugs.

To avoid the "withdrawal" syndrome, stop taking the medication gradually, reducing the dosage to a minimum.

When taking sleeping pills, the patient may have anterograde amnesia. As a rule, it manifests itself in the interruption of sleep, and after a long time between taking the medication and going to sleep.

To reduce such risks, it is necessary:

  • Ensure a sleep duration of at least 6 hours;
  • Take medicine right before bedtime.

This medication is not indicated for depression therapy. He can mask her symptoms.

An effective and safe dose of "Relaxon" in children and adolescents under 18 years old has not been established by specialists. Therefore, taking the drug at this age is prohibited.

Due to the pharmacological properties of the hypnotic, it can have an adverse effect on a patient's ability to drive vehicles, as well as engage in hazardous activities that require increased attention and quick response. In this regard, during the treatment with this drug should be extremely cautious.

Sleeping pills "Relaxon": price and analogy

What can replace the drug "Relaxon"? This drug has many analogues. The most effective are the following medicines: Milovan, Imovan, Thorson, Somnol, Slipwell, Zolinox, Piklodorm, Zopiclone.

All these drugs, including "Relaxon", are dispensed in pharmacies only on prescription. As for the price, this means it is not very high. 20 tablets of sleeping pills (7.5 mg) can be purchased for 120-160 rubles.

Reviews of sleeping pills

According to specialists, the drug "Relaxon" is a sleeping drug of the third generation. By the way, they include Zaleplon and Zolpidem. These drugs are highly effective and absolutely safe.

Patients report that after taking sleeping pills, their sleep quality has improved markedly. At the same time, the fast-phase sleep, necessary for restoring the psychoemotional state, was completely preserved.

This drug has a good effect on the slow-wave phase of sleep, which is extremely important for the physical recovery of the human body.

According to specialists, this drug contributes to the normalization of the structure of sleep in all types of disorders. At the same time, it has the least likelihood of addiction.

The patients' testimonies indicate that the sleeping pills "Relaxon" are well tolerated, without having any effect on the person's daily activity. However, doctors do not recommend taking this medicine at their discretion. The patient should always consult a doctor and follow all the recommended dosages.

Similar articles

 

 

 

 

Trending Now

 

 

 

 

Newest

Copyright © 2018 en.birmiss.com. Theme powered by WordPress.